Assistant Professor Dr. / Bassem Heshmat Naguib
Pharmaceutical Organic Chemistry
bassem.naguib@pharma.cu.edu.eg
Latest List of Publications
1- “Design and Novel Synthetic Approach Supported with Molecular Docking and Biological Evidence for Naphthoquinone-Hydrazinotriazolothiadiazine Analogs as Potential Anticancer Inhibiting Topoisomerase-IIB” Bioorganic Chemistry Vol 96, 103641 (2020). Samy Mohamady, Mahmoud Salama Ahmed, Abdullah Gibriel, Moataz S. Hendy and Bassem H. Naguib.
2- “Structure-based drug design, synthesis, In vitro, and In vivo biological evaluation of indole-based biomimetic analogs targeting estrogen receptor-α inhibition” European Journal of Medicinal Chemistry Vol 166, 281-290 (2019). Moataz S. Hendy, Aya A. Ali, Lubna Ahmed, Reham Hossam, Alaa Mostafa, Mohamed M. Elmazar, Bassem H. Naguib, Yasmeen M. Attia, Mahmoud Salama Ahmed.
3- “Design, Synthesis, Cytotoxic Activity and Apoptosis-inducing Action of Novel Cinnoline Derivatives as Anticancer Agents.” Anti-Cancer Agents in Medicinal Chemistry Vol 18 (8), 1208 - 1217 (2018), Manal M. Kandeel, Aliaa M. Kamal, Bassem H. Naguib and Marwa S. A. Hassan
4- “Synthesis of New Pyridothienopyrimidinone and Pyridothienotriazolopyrimidine Derivatives as Pim-1 Inhibitors.” Journal of Enzyme Inhibition and Medicinal Chemistry Vol 33(1), 58-66 (2018), Hala B. El-Nassan, Bassem H. Naguib, Engy A. Beshay
5- “Synthesis of new pyridothienopyrimidinone derivatives as Pim-1 inhibitors.” Journal of Enzyme Inhibition and Medicinal Chemistry Vol 32(1), 457-467 (2017), Bassem H. Naguib, Hala B. El-Nassan, Abdelghany, T.M.
6- “Synthesis of new thieno[2,3-b]pyridine derivatives as pim-1 inhibitors.”, Journal of Enzyme Inhibition and Medicinal Chemistry Vol 31(6), 1718-1725 (2016), Bassem H. Naguib, Hala B. El-Nassan.
7- “Synthesis and anticonvulsant activity of new phenytoin derivatives.” European Journal of Medicinal Chemistry Vol 60, 57-63(2013). Samir Botros Salib, Nadia Abdalla Khalil, Bassem H. Naguib, Yara Sayed El-Dash.
8- “Phenytoin-based Bivalent Ligands: Design, Synthesis and anticonvulsant Activity”. Archives of Pharmacal Research Vol 35(12), 2105-2116 (2012). Samir Botros Salib, Nadia Abdalla Khalil, Bassem Heshmat Naguib, Yara Sayed El-Dash
9- “Synthesis and tranquillizing effect of new dibenzoxazepines and pyridobenzoxazepines”, Egyptian Journal of Chemistry Vol 54(6), 691-701 (2011), S. Botros, B. H. Naguib and A. N. Osman
10- “Synthesis and tranquillizing effect of new 1,4-benzoxazepines”, Egyptian Journal of Chemistry Vol 54(5), 565-578 (2011), S. Botros, B. H. Naguib and A. N. Osman
11- “Pyridine carbonitrile derivatives as versatile synthons for some heterocyclic compounds of pharmaceutical interest”, Bulletin of the Faculty of Pharmacy, Cairo University Vol 41 (3) 2003 p.1-11, M. Mohsen Ismail, R. H. Omar, M.M. Said, A. Ahmady, A. H. Omar, B. H. Naguib.